mammal (species unspecified) |
LD50 |
unreported |
1109mg/kg (1109mg/kg) |
|
French Demande Patent Document. Vol. #2454807, |
man |
TDLo |
oral |
1714ug/kg/3D- (1.714mg/kg) |
LUNGS, THORAX, OR RESPIRATION: CYANOSIS
BLOOD: METHEMOGLOBINEMIA-CARBOXYHEMOGLOBIN |
Australian and New Zealand Journal of Medicine. Vol. 27, Pg. 596, 1997. |
mouse |
LD50 |
intramuscular |
1080mg/kg (1080mg/kg) |
|
Drugs in Japan Vol. 6, Pg. 72, 1982. |
mouse |
LD50 |
intraperitoneal |
720mg/kg (720mg/kg) |
|
Yakkyoku. Pharmacy. Vol. 24, Pg. 431, 1973. |
mouse |
LD50 |
intravenous |
> 40mg/kg (40mg/kg) |
BEHAVIORAL: ATAXIA
SKIN AND APPENDAGES (SKIN): HAIR: OTHER |
Kiso to Rinsho. Clinical Report. Vol. 19, Pg. 4947, 1985. |
mouse |
LD50 |
oral |
1050mg/kg (1050mg/kg) |
|
Drugs in Japan Vol. 6, Pg. 72, 1982. |
mouse |
LD50 |
subcutaneous |
1050mg/kg (1050mg/kg) |
|
Drugs in Japan Vol. 6, Pg. 72, 1982. |
rabbit |
LD50 |
intravenous |
> 40mg/kg (40mg/kg) |
BEHAVIORAL: SOMNOLENCE (GENERAL DEPRESSED ACTIVITY)
BEHAVIORAL: ATAXIA |
Kiso to Rinsho. Clinical Report. Vol. 19, Pg. 4947, 1985. |
rat |
LD50 |
intramuscular |
> 2gm/kg (2000mg/kg) |
|
Drugs in Japan Vol. 6, Pg. 72, 1982. |
rat |
LD50 |
intraperitoneal |
670mg/kg (670mg/kg) |
SENSE ORGANS AND SPECIAL SENSES: PTOSIS: EYE
LUNGS, THORAX, OR RESPIRATION: RESPIRATORY DEPRESSION
BEHAVIORAL: CHANGES IN MOTOR ACTIVITY (SPECIFIC ASSAY) |
Oyo Yakuri. Pharmacometrics. Vol. 35, Pg. 287, 1988. |
rat |
LD50 |
intravenous |
> 40mg/kg (40mg/kg) |
BEHAVIORAL: SOMNOLENCE (GENERAL DEPRESSED ACTIVITY)
BEHAVIORAL: ATAXIA |
Kiso to Rinsho. Clinical Report. Vol. 19, Pg. 4947, 1985. |
rat |
LD50 |
oral |
747mg/kg (747mg/kg) |
|
Gekkan Yakuji. Pharmaceuticals Monthly. Vol. 26, Pg. 309, 1984. |
rat |
LD50 |
skin |
> 3gm/kg (3000mg/kg) |
|
Oyo Yakuri. Pharmacometrics. Vol. 35, Pg. 287, 1988. |
rat |
LD50 |
subcutaneous |
1237mg/kg (1237mg/kg) |
BEHAVIORAL: CONVULSIONS OR EFFECT ON SEIZURE THRESHOLD
BEHAVIORAL: EXCITEMENT |
Yakuri to Chiryo. Pharmacology and Therapeutics. Vol. 10, Pg. 2109, 1982. |
women |
TDLo |
oral |
100ug/kg (0.1mg/kg) |
BEHAVIORAL: COMA
CARDIAC: PULSE RATE
CARDIAC: OTHER CHANGES |
Southern Medical Journal. Vol. 84, Pg. 369, 1991.
|